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Alogliptin Benzoate

  (SYR 322)
目录号: PC-99030

Alogliptin Benzoate (SYR-322) 是一种有效的、具有选择性口服活性的 DPP-4 的抑制剂

CAS NO.:850649-62-6

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规格 价格 库存
10mg 850.00 现货
50mg 3000.00 现货
100mg 4200.00 现货

基本信息

Alogliptin is an orally bioavailable dipeptidyl peptidase 4 (DPP-4) inhibitor (IC50 = 6.9 nM) that is selective for DPP-4 over DPP-2, DPP-8, DPP-9, prolyl endopeptidase, fibroblast activation protein (FAP), and tryptase (IC50s = >100,000 nM).It does not inhibit cytochrome P450 enzymes and does not block the human ether-a-go-go-related gene (hERG) channel when used at concentrations up to 30 μM.2 Alogliptin inhibits DPP-4 activity in vivo in rats, dogs, and cynomolgus monkeys (EC50s = 3.4, 4.9, and 5.6 ng/ml, respectively, in plasma).

CAS 850649-62-6
分子量 461.51
分子式

C25H27N5O4

溶剂

DMSO

纯度 98%
存储温度 -20℃

相关说明文档

储备液配置

浓度 体积 质量
1mg 5mg 10mg
1 mM 2.1668 mL 10.8340 mL 21.6680 mL
5 mM 0.4334 mL 2.1668 mL 4.3336 mL
10 mM 0.2167 mL 1.0834 mL 2.1668 mL
注:请根据所选浓度进行配置储备液,配置好储备液后进行分装低温保存,避免反复冻融!PCM提供多种溶剂,如:DMSO(PC-57930);玉米油(PC-86094);棉籽油(PC-30875)等

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