AM281
AM281 是一种选择性 CB1 受体拮抗剂
CAS NO.：202463-68-1
| 规格 | 价格 | 库存 |
|---|---|---|
| 5mg | 800.00 | 现货 |
| 10mg | 1250.00 | 现货 |
| 50mg | 4000.00 | 现货 |
基本信息
|
AM281 is a potent and selective central cannabinoid (CB1) receptor antagonist/inverse agonist (Kis = 12 nM and 4,200 nM for CB1 and CB2, respectively).Structurally, it is an analog of the CB1 inverse agonist rimonabant (Cat No. PC-55667). It has no effect on the vanilloid TRPV1 receptor.AM281 has been used to evaluate the potential effects of compounds at CB1.It has also been used to study the membrane localization and cycling of CB1. |
|
| CAS | 202463-68-1 |
| 分子量 | 557.21 |
| 分子式 |
C21H19Cl2lN4O2 |
| 溶剂 | DMSO/DMF |
| 纯度 | 98% |
| 存储温度 | -20℃ |
相关说明文档
储备液配置
|
浓度
体积
质量
|
1mg | 5mg | 10mg |
| 1 mM | 1.7947 mL | 8.9733 mL | 17.9466 mL |
| 5 mM | 0.3589 mL | 1.7947 mL | 3.5893 mL |
| 10 mM | 0.1795 mL | 0.8973 mL | 1.7947 mL |
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