Hemopressin (human, mouse)
Selective CB1 inverse agonist。(Pro-Val-Asn-Phe-Lys-Leu-Leu-Ser-His/PVNFKLLSH)
CAS NO.:1314035-51-2
规格 | 价格 | 库存 |
---|---|---|
1mg | 2560.00 | 现货 |
2mg | 3890.00 | 现货 |
5mg | 8990.00 | 现货 |
基本信息
Bioactive endogenous peptide substrate for endopeptidase 24.15 (ep24.15), neurolysin (ep24.16) and ACE. Ki values are 27.76, 3.43 and 1.87 μM respectively. Potent hypotensive in vivo. Also acts as a selective CB1 receptor inverse agonist. Displays antinociceptive activity in vivo. |
|
CAS | 1314035-51-2 |
分子量 | 1054.24 |
分子式 |
C50H79N13O12 |
溶剂 |
H2O |
纯度 | 98% |
存储温度 | -20℃ |
相关说明文档
储备液配置
浓度
体积
质量
|
1mg | 5mg | 10mg |
1 mM | 0.9486 mL | 4.7428 mL | 9.4855 mL |
5 mM | 0.1897 mL | 0.9486 mL | 1.8971 mL |
10 mM | 0.0949 mL | 0.4743 mL | 0.9486 mL |
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