Imperatorin
Imperatorin 是 TRPV1 的微弱激动剂
CAS NO.：482-44-0
| 规格 | 价格 | 库存 |
|---|---|---|
| 10mg | 500.00 | 现货 |
| 20mg | 950.00 | 现货 |
| 50mg | 1700.00 | 现货 |
基本信息
|
Imperatorin is an effective of NO synthesis inhibitor (IC50=9.2 μmol), which also is a BChE inhibitor (IC50=31.4 μmol); it is a weak agonist of TRPV1 with EC50 of 12.6±3.2 μM. Imperatorin is a potent myorelaxant agent and acts as a calcium antagonist on vascular smooth muscle. Imperatorin has anticonvulsant, anti-inflammatory, anti-oxidant, neuroprotection, and anti-cancer effects, it also has been used in herbal formulations for the treatment of hypertension and cardiovascular diseases. Imperatorin dampens neuronal excitability by inhibiting voltage-gated Na + channels (VGSC), and blocks the HSP27 and HSP72 gene expression. |
|
| CAS | 482-44-0 |
| 分子量 | 270.28 |
| 分子式 |
C16H14O4 |
| 溶剂 | DMSO |
| 纯度 | 98% |
| 存储温度 | -20℃ |
相关说明文档
储备液配置
|
浓度
体积
质量
|
1mg | 5mg | 10mg |
| 1 mM | 3.6999 mL | 18.4993 mL | 36.9987 mL |
| 5 mM | 0.7400 mL | 3.6999 mL | 7.3997 mL |
| 10 mM | 0.3700 mL | 1.8499 mL | 3.6999 mL |
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